Agmatine

A metabolite of arginine that may support mood, pain, and athletic performance.

Also known as: (4-aminobutyl)guanidine

other Names
(4-aminobutyl)guanidine
primary Benefits
Mood support, pain relief, athletic performance
common Dose
500-1000 mg per day
best Form
Sulfate salt in capsules or powder
timing
30-60 minutes before workouts or as needed for other benefits
safety Rating
Moderate Caution

Overview

Agmatine is a compound that is naturally produced in the body from the amino acid arginine. It is found in various tissues and is thought to act as a neurotransmitter and neuromodulator. Agmatine has been studied for a wide range of potential benefits, including its ability to support mood, reduce pain, and enhance athletic performance. It is believed to work through multiple mechanisms, including its interaction with various receptors in the brain, its ability to modulate nitric oxide production, and its antioxidant properties. Research on agmatine is still in its early stages, but some studies suggest that it may be beneficial for conditions such as depression, neuropathic pain, and drug addiction. It has also gained popularity in the fitness community as a pre-workout supplement, with claims that it can improve muscle pumps and endurance. However, more research is needed to confirm these effects and to determine the optimal dosage and long-term safety of agmatine supplementation.

Key Benefits

May Improve Mood

Agmatine may have antidepressant-like effects by modulating various neurotransmitter systems in the brain.

May Reduce Pain

Some studies suggest that agmatine can help alleviate neuropathic pain by interacting with pain pathways.

May Enhance Athletic Performance

Agmatine may improve muscle pumps and endurance by increasing nitric oxide production.

Dosage & How to Take

Start with a low dose and assess tolerance. Consult with a healthcare professional before use.

PurposeDoseNotes
Mood Support500-1000 mg per dayMay be taken in divided doses.
Pain Relief1000-2670 mg per dayHigher doses may be needed for this purpose.
Athletic Performance500-1000 mgTake 30-60 minutes before exercise.

Best Time to Take

For athletic performance, take before workouts. For other benefits, it can be taken at any time of day.

With or Without Food

Can be taken with or without food.

Forms & Bioavailability

FormAbsorptionBest ForNotes
Agmatine SulfateHighGeneral useThe most common form of agmatine supplement.

Side Effects & Safety

Common

  • Nausea
  • Diarrhea
  • Stomach upset

Rare

  • Headache
  • Dizziness

Contraindications

  • Individuals with kidney or liver disease should use with caution.

Interactions

Blood pressure medicationModerate

May enhance the effects of these medications

ArginineMild

May compete for absorption

Scientific Research

2010Pharmacological Reports

Agmatine enhances the antidepressant-like effects of selective serotonin reuptake inhibitors in mice

Agmatine may be a useful adjunct to antidepressant therapy.

2014Pain Physician

Agmatine: a potential novel therapeutic agent for neuropathic pain

A review of studies suggesting agmatine may be effective in treating neuropathic pain.

Food Sources

Fermented foods
Wine
Beer

Products With Agmatine

6 products in our database contain this ingredient

Frequently Asked Questions

Medical Disclaimer

This content is for educational and informational purposes only and is not intended as medical advice. Always consult with a qualified healthcare professional before starting any supplement regimen, especially if you have pre-existing health conditions or are taking medications. The statements on this page have not been evaluated by the Food and Drug Administration.